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Search Results for " gonadotropin releasing hormone receptor "

20

Compounds

Cat No. Product Name Synonyms Targets
TP1288 Fertirelin Others
Fertirelin, or fertirelin acetate, sold under the brand name Ovalyse, is a gonadotropin-releasing hormone agonist (GnRH agonist).
T1494 Alarelin Acetate Alarelin GNRH Receptor
Alarelin Acetate is a synthetic GnRH agonist which can directly inhibit proliferation and DNA synthesis of rat GSMC through GnRH receptors.
T5520 Cetrorelix Acetate Cetrorelix GNRH Receptor
Cetrorelix Acetate is gonadotropin-releasing hormone (GnRH) receptor antagonist with an IC50 of 1.21 nM.
T27837 Linzagolix GNRH Receptor
Linzagolix is a small-molecule, non-peptide, orally active gonadotropin-releasing hormone antagonist (GnRH antagonist) which is under development by Kissei Pharmaceutical and ObsEva for the treatment of uterine fibroids,...
T4102 Goserelin acetate Fertilan,ICI-118630 acetate,Zoladex Apoptosis , GNRH Receptor
Goserelin acetate (Fertilan) is a synthetic long-acting agonist of gonadotropin-releasing hormone, used in treatments of cancer.
T11174 (R)-Elagolix NBI-56418 GNRH Receptor
(R)-Elagolix (NBI-56418) is a short-acting, nonpeptide, GnRH antagonist with an IC50 and Ki of 0.25 and 3.7 nM, respectively. administered orally, that unlike injectable depot GnRH agonists and antagonists, produces a do...
T5031 Elagolix sodium NBI-56418 sodium GNRH Receptor
Elagolix sodium (NBI-56418 sodium) is a GnRH receptor (GnRHR) antagonist ( IC50 and Ki of 0.25 and 3.7 nM, respectively).
T10217L Abarelix R3827,PPI 149 GNRH Receptor
Abarelix (PPI 149) is a potent gonadotrophin-releasing hormone (GnRH) antagonist, which is used for prostate cancer treatment.
T3630 Relugolix RVT-601,TAK-385 GNRH Receptor
Relugolix (RVT-601) is an orally available, non-peptide gonadotropin-releasing hormone (GnRH or luteinizing hormone-releasing hormone (LHRH)) antagonist, with potential antineoplastic activity. Relugolix competitively bi...
T5520L Cetrorelix diacetate NS-75A,SB-075 acetate,SB-075 diacetate,Cetrorelix acetate,NS-75A diacetate GNRH Receptor
Cetrorelix diacetate (NS-75A) is is a gonadotropin-releasing hormone antagonist. It works by blocking the action of GnRH upon the pituitary, thus rapidly suppressing the production and action of luteinizing hormone (LH) ...
T21308 Histrelin Supprelin LA,Histrelin Acetate Others
Histrelin (Supprelin LA) acetate is a nonapeptide analog of gonadotropin-releasing hormone (GnRH) with added potency. It is considered a GnRH agonist. Histrelin is used in the treatment of hormone-sensitive cancers of th...
T10988L Degarelix acetate(214766-78-6 free base) GNRH Receptor
Degarelix acetate is a competitive and reversible antagonist of gonadotropin-releasing hormone receptor (GnRHR) .
TP2337 Ganirelix Acetate GNRH Receptor
Ganirelix Acetate is a gonadotropin-releasing hormone (GnRH) receptor antagonist
TP1307 Buserelin Acetate (57982-77-1 free base) Buserelin Acetate GNRH Receptor
Buserelin Acetate (57982-77-1 free base) (Buserelin Acetate) is an agonist of gonadotropin-releasing hormone receptor(GnRHR).
T23412 T 98475 Others
gonadotropin-releasing hormone (GnRH, LHRH) receptor antagonist,orally active
T17301 Opigolix Others
Opigolix is a Gonadotropin-releasing hormone receptor antagonist.
T10988 Degarelix GNRH Receptor
Degarelix is a competitive and reversible gonadotropin-releasing hormone receptor (GnRHR) antagonist.
T10475 BAY-784 Others
BAY-784 is a gonadotropin-releasing hormone receptor (GnRH-R) antagonist (IC50s: 21 and 24 nM for human and rat GnRH-R).
T76351 [D-Ala6]-LH-RH
[D-Ala6]-LH-RH, a Luteinizing-hormone-releasing hormone (LHRH) analogue, functions as a gonadotropin-releasing hormone (GnRH) receptor agonist [1].
TP1936 RFRP-3(human) RFRP 3 (human)
Agonist of the NPFF1 receptor (IC50 = 0.7 nM for inhibition of forskolin-induced cAMP production). Homolog of gonadotropin-inhibitory hormone (GnIH); inhibits activity of gonadotropin-releasing hormone (GnRH) neurons.
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TargetMol